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  1. ̾¾Î

    ʬÎà

    µ¡½ø

    from PMDA, ¿³ººÊó¹ð(1)(rev. Ê¿À®21ǯ3·î17Æü) (in vitro)

    (Âå¼Õʪ, N-æ¥á¥Á¥ëÂÎ)

    (Âå¼Õʪ, 8-¥Ò¥É¥í¥­¥·ÂÎ)

    (Âå¼Õʪ, 8-¥Ò¥É¥í¥­¥·-N-æ¥á¥Á¥ëÂÎ)

    (Âå¼Õʪ, N-»À²½ÂÎ)

    (Âå¼Õʪ, N-æ¥á¥Á¥ëÂΤÎβ»ÀÊú¹çÂÎ)


    from ['¥ì¥á¥í¥ó'] IF ¥·¥§¥ê¥ó¥°¡¦¥×¥é¥¦³ô¼°²ñ¼Ò (rev.1 2009ǯ7·î) (in vitro)

    (Âå¼Õʪ, N-æ¥á¥Á¥ëÂÎ)


    from PMDA, ['¥ê¥Õ¥ì¥Ã¥¯¥¹'] ÌÀ¼£À½²Û³ô¼°²ñ¼Ò (rev.1 2009ǯ7·î)

    (Âå¼Õʪ, N-æ¥á¥Á¥ëÂÎ)


    from DailyMed, ['remeron'] Organon USA, Inc. (rev. 08/2008)


    from KEGG


    from eMC, ['zispin'] Organon Laboratories Limited (rev. 07/03/2006)

    ¹ÚÁÇ

    Á˳²

    from PMDA, ¿³ººÊó¹ð(1)(rev. Ê¿À®21ǯ3·î17Æü)
    "Î×¾²ºÇÂçÍÑÎÌ¡Ê45 mg¡Ë¤òÅêÍ¿¤·¤¿ºÝ¤Î¸ÄÊ̾ÉÎã¤Ë¤ª¤±¤ëCmax ¤ÎºÇÂçÃÍ¡Ê0.99 ¦Ìmol/L¡Ë"
    "Î×¾²¾åÌäÂê¤È¤Ê¤ë²ÄǽÀ­¤ÏÄ㤤", ­¶¡¥£´¡¥¡Êüò¡Ë ¡ãÄó½Ð¤µ¤ì¤¿»ñÎÁ¤Î³µÎ¬¡ä ¡Ê£±¡Ë.

    ¹ÚÁÇKiÃÍ [¦Ìmol/L]
    CYP2D641.1
    CYP1A2159
    CYP3A4210


    from PMDA, ['¥ê¥Õ¥ì¥Ã¥¯¥¹'] ÌÀ¼£À½²Û³ô¼°²ñ¼Ò (rev.1 2009ǯ7·î)

    from eMC, ['zispin'] Organon Laboratories Limited (rev. 07/03/2006)

    • (CYP1A2) (in virto) "very weak"
    • (CYP2D6) (in virto) "very weak"
    • (CYP3A) (in virto) "very weak"


    ͶƳ

    from PMDA, ¿³ººÊó¹ð(1)(rev. Ê¿À®21ǯ3·î17Æü)
    "µ¡¹½¤Ï¡ÊÃæÎ¬¡Ë ¥Ò¥È¤Ç¤Î±Æ¶Á¤Ë¤Ä¤¤¤Æ¤Ï¡¢Î×¾²»î¸³À®ÀÓ¤òƧ¤Þ¤¨¤ÆÈ½ÃǤ¹¤ëɬÍפ¬¤¢¤ë¤È¹Í¤¨¤ë¡£", ­¶¡¥£³¡¥¡Êüò¡Ë ¡ã¿³ºº¤Î³µÎ¬¡ä ¡Ê£²¡Ë.


    Âå¼Õ

    from PMDA, ¿³ººÊó¹ð(1)(rev. Ê¿À®21ǯ3·î17Æü)

    from PMDA, ['¥ê¥Õ¥ì¥Ã¥¯¥¹'] ÌÀ¼£À½²Û³ô¼°²ñ¼Ò (rev.1 2009ǯ7·î)

    from DailyMed, ['remeron'] Organon USA, Inc. (rev. 08/2008)

    Ê»ÍѶش÷¡¦Ãí°Õ

    from PMDA, ['¥ê¥Õ¥ì¥Ã¥¯¥¹'] ÌÀ¼£À½²Û³ô¼°²ñ¼Ò (rev.1 2009ǯ7·î)


    from DailyMed, ['remeron'] Organon USA, Inc. (rev. 08/2008)


    from eMC, ['zispin'] Organon Laboratories Limited (rev. 07/03/2006)

    µ¬À©¶èʬ

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    • afloyan
    • avanza
    • azapin
    • depreram
    • rexer
    • vastat

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